- Dextroamphetamine (approved / labelled) - stimulant
- Lisdexamfetamine (approved / labelled) - stimulant
- Mecasermin / Recombinant Human IGF-1 (approved / labelled) - doping
- Methylphenidate (approved / labelled) - stimulant
- Nandrolone Decanoate (approved / labelled) - doping
- Oxandrolone (approved / labelled) - doping
- Oxymetholone (approved / labelled) - doping
- Racemic Amphetamine Sulfate (approved / labelled) - stimulant
- Dehydroepiandrosterone (human RCT) - doping
- Ephedrine (human RCT) - stimulant
- Methandienone (human RCT) - doping
- Oral Salbutamol (human RCT) - doping
- PEG-MGF / Pegylated Mechano Growth Factor (human RCT) - doping
- Yohimbine (human RCT) - stimulant
- Clenbuterol (early human) - doping, stimulant
- Follistatin / FS344 (early human) - doping
- Ligandrol (early human) - doping
- RAD140 (early human) - doping
- Stanozolol (early human) - doping
- AC-262536 (preclinical) - doping
- Andarine (preclinical) - doping
- Dermorphin (preclinical) - doping
- IGF-1 LR3 / DES(1-3)IGF-1 (preclinical) - doping
- LGD-3303 (preclinical) - doping
- S-23 (preclinical) - doping
- Trenbolone (preclinical) - doping
- Ursolic Acid (preclinical) - skeptical priority
- YK11 (preclinical) - doping
- ACP-105 (mechanistic) - doping, toxicology