- (-)-BPAP (preclinical)
- 5-Amino-1MQ (preclinical)
- 522-054 (preclinical)
- AC-262536 (preclinical)
- ACE-031 (human RCT)
- ACE-167 (preclinical)
- ACP-105 (mechanistic)
- Adamax (mechanistic)
- AHK-Cu (mechanistic)
- Amlodipine (approved / labelled)
- Andarine (preclinical)
- AOD9604 (early human)
- Apitegromab (early human)
- ARA-290 / Cibinetide (early human)
- Arginine (preclinical)
- Astaxanthin (preclinical)
- Astaxanthin-fortified yogurt (mechanistic)
- ATR-258 (early human)
- Baicalin (preclinical)
- Batatasin III (preclinical)
- Bazedoxifene (approved / labelled)
- Berberine (human RCT)
- Bergamot Phytosome (human RCT)
- Betulinic Acid (mechanistic)
- Bilirubin / Biliverdin axis (mechanistic)
- Bimagrumab (human RCT)
- BMS-564929 (preclinical)
- BPC-157 (preclinical)
- Bremelanotide (approved / labelled)
- Cagrilintide (human RCT)
- Cagrilintide + Semaglutide / CagriSema (human RCT)
- Carnosine / Beta-Alanine (human RCT)
- Cartalax (preclinical)
- Cerebrolysin (human RCT)
- Cetoleic Acid Concentrate (human RCT)
- Citrulline / L-Citrulline (human RCT)
- CJC-1295 (early human)
- CJC-1295 No DAC / Modified GRF(1-29) (early human)
- Clenbuterol (early human)
- Clomiphene (approved / labelled)
- Clomipramine (approved / labelled)
- Clonidine (approved / labelled)
- Clorgyline (mechanistic)
- Corylin (preclinical)
- Creatine (human RCT)
- Cutamesine (early human)
- CVN424 (human RCT)
- Damiana Extract (mechanistic)
- Declozindol (unresolved)
- Dehydroepiandrosterone (human RCT)
- Dehydroevodiamine HCl (preclinical)
- Delta Sleep-Inducing Peptide (early human)
- Dermorphin (preclinical)
- Dexmedetomidine (approved / labelled)
- Dextroamphetamine (approved / labelled)
- Dieckol (preclinical)
- Dihexa (preclinical)
- Diphenhydramine (approved / labelled)
- Doxycycline (human RCT)
- Elunetirom (early human)
- Enclomiphene (human RCT)
- Enobosarm (human RCT)
- Ephedrine (human RCT)
- Epitalon / Epithalon (preclinical)
- Esmirtazapine (human RCT)
- Eucommia ulmoides Leaf Extract (preclinical)
- EUK-134 (early human)
- Everolimus (approved / labelled)
- Fenfluramine (approved / labelled)
- Finasteride (approved / labelled)
- Flecainide (approved / labelled)
- Follistatin / FS344 (early human)
- Forsythoside A (preclinical)
- FOXO4-DRI (preclinical)
- Galactooligosaccharides / RP-G28 (human RCT)
- Garetosmab (human RCT)
- Gellan Gum (preclinical)
- GHK (mechanistic)
- GHK-Cu (mechanistic)
- GHRP-2 / Pralmorelin (early human)
- GHRP-6 (early human)
- Glutamine / L-Glutamine (approved / labelled)
- Glutathione (human RCT)
- Gonadorelin (early human)
- GSK2881078 (early human)
- Gynostemma pentaphyllum Extract (human RCT)
- Hexarelin (early human)
- High-Molecular-Weight Hyaluronic Acid (preclinical)
- HMB (human RCT)
- HMG / Menotropins (approved / labelled)
- Human chorionic gonadotropin (approved / labelled)
- Human Growth Hormone / Somatropin (approved / labelled)
- Hyaluronic Acid / Sodium Hyaluronate (human RCT)
- Hydroxyzine (approved / labelled)
- Ibutamoren (human RCT)
- IGF-1 LR3 / DES(1-3)IGF-1 (preclinical)
- Imidazenil (preclinical)
- INT131 (early human)
- Ipamorelin (early human)
- Irdabisant (preclinical)
- Keraxidil (unresolved)
- Kisspeptin-10 (early human)
- KPV (preclinical)
- L-carnitine (human RCT)
- Lemon Myrtle Extract (human RCT)
- Leonurine (preclinical)
- Leucine (human RCT)
- LGD-3303 (preclinical)
- Ligandrol (early human)
- Lisdexamfetamine (approved / labelled)
- LL-37 (human RCT)
- M40401 (preclinical)
- Maslinic Acid (human RCT)
- Mazdutide (human RCT)
- Mecasermin / Recombinant Human IGF-1 (approved / labelled)
- Metformin (approved / labelled)
- Methandienone (human RCT)
- Methylphenidate (approved / labelled)
- Mexidol (mechanistic)
- Milk Kefir (human RCT)
- Mirabegron (approved / labelled)
- MOTS-c (preclinical)
- NAD+ / Intravenous NAD (early human)
- NADH (human RCT)
- Nandrolone Decanoate (approved / labelled)
- Nebivolol (approved / labelled)
- Nicotinamide Mononucleotide (human RCT)
- Nicotinamide Riboside (human RCT)
- Oleracein E (preclinical)
- Oral Salbutamol (human RCT)
- Oroxylin A (preclinical)
- Ospemifene (approved / labelled)
- Oxandrolone (approved / labelled)
- Oxymetholone (approved / labelled)
- Oxytocin (approved / labelled)
- P21 / P021 Peptide (preclinical)
- Paeonol (mechanistic)
- PDE5 inhibitors / Cialis / Viagra (approved / labelled)
- PE-22-28 (preclinical)
- PEG-MGF / Pegylated Mechano Growth Factor (human RCT)
- Pemafibrate (human RCT)
- Phosphatidic Acid (human RCT)
- Phycocyanobilin / Spirulina (human RCT)
- Piceatannol (human RCT)
- Pinealon (early human)
- Piperlongumine (preclinical)
- Polydatin (preclinical)
- Protein Supplementation (human RCT)
- Racemic Amphetamine Sulfate (approved / labelled)
- RAD140 (early human)
- Raloxifene (approved / labelled)
- Rapamycin / Sirolimus (approved / labelled)
- Retatrutide (human RCT)
- RTB101 (human RCT)
- S-23 (preclinical)
- Saskatoon Berry (early human)
- SC19 MC4R agonist lead (preclinical)
- Schisandrin B (preclinical)
- Sciadonic Acid (preclinical)
- Seladelpar (approved / labelled)
- Selank (early human)
- Selegiline (approved / labelled)
- Semaglutide (approved / labelled)
- Semax (early human)
- Sermorelin (early human)
- Sertraline (approved / labelled)
- Setmelanotide (approved / labelled)
- Sildenafil / Viagra (approved / labelled)
- SLU-PP-332 (preclinical)
- SNAP-8 / Acetyl Octapeptide-3 (early human)
- Spilanthes acmella Extract (preclinical)
- SR-17018 (preclinical)
- SS-31 / Elamipretide (approved / labelled)
- Stanozolol (early human)
- Survodutide (human RCT)
- Tadalafil / Cialis (approved / labelled)
- Tamoxifen (approved / labelled)
- TB-500 / thymosin beta-4-related products (human RCT)
- Telmisartan (approved / labelled)
- Tesamorelin (approved / labelled)
- Testosterone (approved / labelled)
- THN102 (human RCT)
- Thymalin (early human)
- Thymosin alpha-1 (human RCT)
- Tirzepatide (approved / labelled)
- Toremifene (approved / labelled)
- Trazodone (approved / labelled)
- Trenbolone (preclinical)
- Trevogrumab (human RCT)
- Tribulus cistoides Extract (preclinical)
- Trigonelline (preclinical)
- Ursolic Acid (preclinical)
- VIP / Vasoactive Intestinal Peptide (early human)
- Vitamin B12 / Cobalamin (approved / labelled)
- Vitamin C / Ascorbic Acid (human RCT)
- Vitamin D / D3 (human RCT)
- Vornorexant (human RCT)
- Water Kefir (mechanistic)
- YK11 (preclinical)
- Yohimbine (human RCT)