- Clomiphene (approved / labelled) - testosterone
- Dextroamphetamine (approved / labelled) - stimulant
- Finasteride (approved / labelled) - testosterone
- Human chorionic gonadotropin (approved / labelled) - testosterone
- Human Growth Hormone / Somatropin (approved / labelled) - growth hormone
- Lisdexamfetamine (approved / labelled) - stimulant
- Mecasermin / Recombinant Human IGF-1 (approved / labelled) - doping, growth hormone
- Methylphenidate (approved / labelled) - stimulant
- Nandrolone Decanoate (approved / labelled) - androgen therapy, doping, steroid
- Oxandrolone (approved / labelled) - doping, steroid
- Oxymetholone (approved / labelled) - doping, steroid
- Racemic Amphetamine Sulfate (approved / labelled) - stimulant
- Tesamorelin (approved / labelled) - growth hormone
- Testosterone (approved / labelled) - androgen therapy, steroid, testosterone
- ACE-031 (human RCT) - myostatin
- Bimagrumab (human RCT) - myostatin
- Dehydroepiandrosterone (human RCT) - doping, steroid, testosterone
- Enclomiphene (human RCT) - testosterone
- Enobosarm (human RCT) - SARM
- Ephedrine (human RCT) - stimulant
- Garetosmab (human RCT) - myostatin
- Ibutamoren (human RCT) - SARM adjacent, growth hormone
- Methandienone (human RCT) - doping, steroid
- Oral Salbutamol (human RCT) - doping
- PEG-MGF / Pegylated Mechano Growth Factor (human RCT) - doping, igf axis
- Trevogrumab (human RCT) - myostatin
- Vitamin D / D3 (human RCT) - testosterone
- Yohimbine (human RCT) - stimulant
- Apitegromab (early human) - myostatin
- CJC-1295 (early human) - growth hormone
- CJC-1295 No DAC / Modified GRF(1-29) (early human) - growth hormone
- Clenbuterol (early human) - doping, stimulant
- Follistatin / FS344 (early human) - doping, myostatin
- GHRP-2 / Pralmorelin (early human) - growth hormone
- GHRP-6 (early human) - growth hormone
- GSK2881078 (early human) - SARM
- Hexarelin (early human) - growth hormone
- Ipamorelin (early human) - growth hormone
- Kisspeptin-10 (early human) - testosterone
- Ligandrol (early human) - SARM, doping
- RAD140 (early human) - SARM, doping
- Sermorelin (early human) - growth hormone
- Stanozolol (early human) - doping, steroid
- AC-262536 (preclinical) - SARM, doping
- ACE-167 (preclinical) - testosterone
- Andarine (preclinical) - SARM, doping
- BMS-564929 (preclinical) - SARM, androgen therapy
- Dermorphin (preclinical) - doping
- IGF-1 LR3 / DES(1-3)IGF-1 (preclinical) - doping, growth hormone
- LGD-3303 (preclinical) - SARM, doping
- S-23 (preclinical) - SARM, doping
- Trenbolone (preclinical) - androgen therapy, doping, steroid
- YK11 (preclinical) - SARM, doping, myostatin
- ACP-105 (mechanistic) - SARM, doping