- Amlodipine (approved / labelled) - angina, cardiovascular, hypertension
- Arginine (preclinical) - vascular function
- Astaxanthin (preclinical) - vascular function
- Berberine (human RCT) - cardiometabolic, lipids
- Bergamot Phytosome (human RCT) - cardiovascular health, lipids, visceral fat
- Bilirubin / Biliverdin axis (mechanistic) - cardiovascular health
- Bremelanotide (approved / labelled) - blood pressure
- Cagrilintide + Semaglutide / CagriSema (human RCT) - cardiometabolic
- Cetoleic Acid Concentrate (human RCT) - cardiovascular health, lipids
- Citrulline / L-Citrulline (human RCT) - blood pressure, cardiovascular health, vascular performance
- Clenbuterol (early human) - cardiovascular
- Clonidine (approved / labelled) - blood pressure, cardiovascular
- Dextroamphetamine (approved / labelled) - cardiovascular
- Dieckol (preclinical) - blood pressure, cardiovascular health, endothelial function
- Eucommia ulmoides Leaf Extract (preclinical) - cardiovascular health, endothelial function
- Flecainide (approved / labelled) - arrhythmia
- Gynostemma pentaphyllum Extract (human RCT) - endothelial function
- Hexarelin (early human) - cardiometabolic
- Hydroxyzine (approved / labelled) - cardiovascular
- Leonurine (preclinical) - atherosclerosis, cardiovascular health, lipids
- Lisdexamfetamine (approved / labelled) - cardiovascular
- Maslinic Acid (human RCT) - cardiovascular health
- Methylphenidate (approved / labelled) - cardiovascular
- Nebivolol (approved / labelled) - cardiovascular, hypertension
- Nicotinamide Riboside (human RCT) - cardiovascular health
- Oral Salbutamol (human RCT) - cardiovascular risk
- Paeonol (mechanistic) - cardiovascular health
- PDE5 inhibitors / Cialis / Viagra (approved / labelled) - blood pressure, cardiovascular, endothelial, pulmonary hypertension, vascular
- Pemafibrate (human RCT) - cardiometabolic, triglycerides
- Phycocyanobilin / Spirulina (human RCT) - blood pressure, cardiovascular health, lipids
- Piceatannol (human RCT) - blood pressure
- Racemic Amphetamine Sulfate (approved / labelled) - cardiovascular
- Saskatoon Berry (early human) - blood pressure, cardiovascular health, lipids
- Sciadonic Acid (preclinical) - cardiovascular health, lipids, triglycerides
- Semaglutide (approved / labelled) - cardiometabolic
- Sildenafil / Viagra (approved / labelled) - blood pressure, cardiovascular, endothelial, pulmonary hypertension, vascular
- SS-31 / Elamipretide (approved / labelled) - cardiology
- Tadalafil / Cialis (approved / labelled) - blood pressure, cardiovascular, endothelial, vascular
- Telmisartan (approved / labelled) - cardiometabolic, hypertension, renal
- Tesamorelin (approved / labelled) - visceral fat
- Trazodone (approved / labelled) - cardiovascular
- Trenbolone (preclinical) - cardiovascular
- VIP / Vasoactive Intestinal Peptide (early human) - vascular
- Vitamin C / Ascorbic Acid (human RCT) - blood pressure, cardiovascular, endothelial, vascular
- Vitamin D / D3 (human RCT) - cardiometabolic